Acta Pharm. 59 (2009) 473-482

 

full paper

Short communication

 

An improved procedure for synthesis of some new 1,3-diaryl-2-propen-1-ones using PEG-400 as a recyclable solvent and their antimicrobial evaluation

BHASKAR S. DAWANE*, SHANKARAIAH G. KONDA, BASEER M. SHAIKH and RAGHUNATH B. BHOSALE

bhaskardawane@rediffmail.com, kondasg@rediffmail.com

 

Organic Research Laboratory, Department of Chemistry, Yeshwant Mahavidyalaya, Nanded-431602 (M.S) India

Accepted August 26, 2009

 

A simple and convenient route is described for the synthesis of novel hetero 1,3-diaryl-2-propen-1-ones (chalcones) by using recyclable poly PEG-400 as an alternative reaction solvent. The reaction is clean with excellent yield, shorter reaction time and reduces the use of volatile organic compounds (VOCs). All the synthesized compounds were evaluated for their antimicrobial activities against several pathogenic representatives.

 

Keywords: 1,3-diaryl-2-propen-1-ones, PEG-400, antimicrobial activity