Acta Pharm. 62 (2012) 83-92
Original research paper
Stability studies of chitosan-DNA-FAP-B
nanoparticles for gene delivery to lung epithelial cells
ZOHREH
MOHAMMADI, FARID ABEDIN DORKOOSH, SAMAN HOSSEINKHANI, TINA AMINI, AMIR ABBAS
RAHIMI, ABDOLHOSSEIN ROUHOLAMINI NAJAFABADI and MORTEZA RAFIEE TEHRANI
rafitehr@ams.ac.ir
1 Department
of Pharmaceutics, Faculty of Pharmacy, Tehran University of Medical Sciences,
Tehran, Iran
2 Nanobiotechnology
Research Center, Avicenna Research Institute, ACECR, Tehran, Iran
3 Department of Biochemistry, Faculty of Science,
Tarbiat Modares University, Tehran, Iran
4 Nobleceuticals
Ltd, Birmingham, United Kingdom
5 Nanobiotechnology Department,
Pasteur Institute of Iran, Tehran, Iran
Accepted January 16, 2012
A successful gene delivery system requires efficiency and stability during storage. Stability studies are imperative for nanomedicines containing biotechnological products such as plasmids and targeting peptides. Chitosan-DNA-FAP-B nanoparticles are novel non-viral vectors for specific gene delivery to the lung epithelial cells. In this study, the storage stability of chitosan-DNA-FAP-B nanoparticles at –20, 5 and 24 ºC was examined. Size, zeta potential and transfection efficiency of these nanoparticles in storage were also evaluated. Stability studies showed that chitosan-DNA-FAP-B nanoparticles were stable after 1 month when stored at –20 °C and retained their initial size, zeta potential and transfection efficiency. However, their stability was not desirable at 5 and 24 ºC. Based on these results, it can be concluded that chitosan-DNA-FAP-B nanoparticles can be a promising candidate for gene delivery to lung epithelial cells with good storage stability at –20 ºC during 1 month.
Keywords: chitosan, FAP-B, nanoparticle, stability, gene
delivery